Basic Peptide Information

DICL ID
DICL_Pep_06854
Ion Channel
Voltage gated potassium channel subfamily H member 2
Peptide Function
Inhibitor
Gene Name
KCNH2

Activity Data (nM)

IC50
22 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified

Sequence Information

Peptide Sequence
YCQKWMWTCDSERKCCEGMVCRLWCKKKLW
Peptide UniProt Accession
UniParc
Not available
Peptide Synonyms/Alias
[CHEMBL3318147; BDBM50051088]
Peptide Species
Thrixopelma pruriens (Peruvian green velvet tarantula)
Peptide Name
Beta/omega-theraphotoxin-Tp2a
CAS Number
484598-36-9

Experimental Conditions

pH
Not mention
Holding Potential (mV)
Not mention
Temperature
Not mention
Test Method
Patch-clamping
Test Species
Not specified

Binding Information

Binding Site
Not specified
Binding Site Residue
Not specified

Ion Channel Information

Gene Abbreviation (ABB)
VGKCs
Ion Channel UniProt Accession
Source Organism
Homo sapiens (Human)

References & Disease Information

Disease
Not specified
PubChem CID
URL
Not available
PMID
Patent
Not available